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barbiturique


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Posted

salut, je ne me souviens plus si cela a été mentionné en cours mais les barbituriques sont ils des agonistes ortho ou allostériques du GABA A? merci

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Posted

Salut :), 

 

Les barbituriques (antiépileptiques) sont des modificateurs allostériques (non compétitifs) positifs (PAM) du récepteur GABA A. Ils vont donc renforcer l'effet du GABA. 

 

Bon courage ! 

 

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